An Open-label, Randomized, 2-sequence, 2-period, 2-treatment, 2-part Study to Evaluate the Relative Bioavailability of SAR443820 in Tablet Formulation Versus Capsule Formulation in Fasted Condition (Part 1) and the Food-effect on SAR443820 in Tablet Formulation (Part 2) in Healthy Adult Male and Female Participants

Study Purpose:

Part 1:

This is an open label, balanced randomized, single dose, 2-sequence, 2-period (period 1 and period 2), 2-treatment crossover (between Treatment A and Treatment B for Part 1), study part to determine the relative bioavailability of SAR443820 in tablet formulation versus capsule formulation under fasted conditions.

Two treatments are as follows:

- Treatment A: SAR443820 - tablet formulation in fasted condition

- Treatment B: SAR443820 - capsule formulation in fasted condition Each administration will be a single dose of SAR443820 separated by a wash out of at least 5 days.

Part 2:

This is an open-label, balanced randomized, single dose, 2-sequence, 2-period (period 1 and period 2), 2-treatment crossover (between Treatment C and Treatment D for Part 2) study part to perform a preliminary assessment of the effect of a high-fat meal on pharmacokinetic parameters of single dose of SAR443820 in tablet formulation.

Two treatments are as follows:

- Treatment C: SAR443820 - tablet formulation in fasted condition

- Treatment D: SAR443820 - tablet formulation in fed condition Each administration will be a single dose of SAR443820 separated by a wash out of at least 5 days.

Participants are not allowed to participate in more than one part of the study. In both Parts 1 and 2, the assessment of pharmacokinetic, safety and tolerability are performed at each treatment period at baseline (prior single dosing) up to 48-hour postdosing in healthy adult male and female participants.

Study Status:

Not recruiting

Disease:

Amyotrophic Lateral Sclerosis (Healthy Volunteers)

Study Type:

Interventional

Type of Intervention:

Drug

Intervention Name:

SAR443820

Placebo:

Yes

Phase:

Phase 1

Study Chair(s)/Principal Investigator(s):

Clinical Sciences & Operations, Sanofi

Clinicaltrials.gov ID:

NCT05797701

Neals Affiliated?

No

Coordinating Center Contact Information

Full Study Summary:

Screening period: up to 4 weeks (Day -28 to Day -2). In both Part 1 and Part 2: Period 1: Day -1 to Day 3 and 5 days wash out period. Period 2: Day -1 to Day 3 and until end-of-study visit at Day 6.

Study Sponsor:

Sanofi

Estimated Enrollment:

18

Estimated Study Start Date:

07 / 28 / 2021

Estimated Study Completion Date:

09 / 06 / 2021

Posting Last Modified Date:

04 / 04 / 2023

Date Study Added to neals.org:

04 / 04 / 2023

Accepts healthy volunteers:

Yes

Minimum Age:

18 Years

Maximum Age:

55 Years

Inclusion Criteria:

- Male or female participant must be 18 to 55 years of age inclusive, at the time of signing the informed consent

- Participants who are overtly healthy as determined by medical evaluation including medical history, physical examination, laboratory tests, and cardiac monitoring

- Body weight between 50.0 and 100.0 kg, inclusive, if male, and between 40.0 and 90.0 kg, inclusive, if female, body mass index between 18.0 and 30.0 kg/m^2, inclusive

- All contraceptive use by men and women should be consistent with local regulations regarding the methods of contraception for those participating in clinical studies

- Having given written informed consent prior to undertaking any study-related procedure

Exclusion Criteria:

- Any history or presence of clinically relevant cardiovascular, pulmonary, gastrointestinal, hepatic, renal, metabolic, hematological, neurological, osteomuscular, articular, psychiatric, systemic, ocular, or infectious disease, or signs of acute illness

- Any medication (including St John's Wort) within 14 days before inclusion or within 5 times the elimination half-life or pharmacodynamic half-life of the medication, with the exception of hormonal contraception or menopausal hormone replacement therapy; any non-live Covid-19 vaccine within the last 2 weeks before randomization, any live attenuated vaccine within the last 28 days before randomization and any other non-vaccine biological drugs given within 4 months before randomization

- Positive result for hepatitis B, C or human immunodeficiency virus (HIV)

- Positive result on urine drug screen

- Positive urine alcohol test

- Positive severe acute respiratory syndrom coronavirus 2 (SARS-CoV-2) test

- Any consumption of citrus fruits (grapefruit, orange, etc) or their juices within 5 days before inclusion

The above information is not intended to contain all considerations relevant to a potential participation in a clinical trial.

Prism Research-Site Number:8400001

Saint Paul, Minnesota 55144
United States